reptides / Cerebrolysin

Cerebrolysin

Cerebrolysin is a porcine-brain hydrolysate mixture measured in milliliters, not one defined peptide. In stroke recovery, the 1,070-person CASTA trial was neutral while the 208-person CARS trial improved the day-90 arm-test result. A Cochrane review found no reliable overall functional benefit, and vascular-dementia evidence remains very uncertain.

porcine-brain peptide hydrolysate

  • Porcine-brain protein hydrolysate
  • No single sequence or molecular mass
  • Stroke evidence is mixed with neutral large trials
  • Current studies dose a finished mixture by volume
Identity Stroke evidence Dementia Mechanism Safety Status

What exactly is Cerebrolysin?

Cerebrolysin is a finished porcine-brain protein hydrolysate containing many peptides and free amino acids. It has no single sequence, molecular formula, mass, receptor, or dose in milligrams of one active ingredient.

Composition study · fingerprints, no active moiety

Analytical in vitro study

Seidl LF, Aigner L. Journal of Medicine and Life, 2024.

The study compared chromatographic fingerprints and in vitro activity among porcine-brain hydrolysates using an originator reference. It does not identify one active peptide or show that market products are clinically interchangeable.

Study design
Laboratory analytical comparison
Funding
Originator material was supplied for comparison
Read the original source
EU CTIS · active academic trial and Romanian authorization

EU clinical-trial registry record

EU CTIS 2024-515591-12-00.

The public record describes an authorized 440-person academic trial and identifies Romanian national marketing authorization 4610/2004/03 for the product used. The trial registration does not yet supply a result and the national authorization does not imply US or EU-central approval.

Participants / model
Planned 440-person stroke-recovery population
Treatment
Cerebrolysin within a randomized academic trial
Study design
Authorized prospective clinical-trial registration

Useful for current research and one specific national authorization only.

Read the original source

Does Cerebrolysin improve stroke recovery?

The compound-specific Cochrane review included seven trials with 1,601 participants and found no reliable functional benefit. CASTA’s global endpoint was neutral; the smaller CARS rehabilitation trial was positive; and a small Chinese three-arm trial reported short-term benefit but excluded 24 of 84 randomized participants without explaining why.

Key stroke evidence
SourceDenominatorFunctional result
Cochrane 20207 trials, 1,601 peopleNo clear clinical benefit; no poolable poor-outcome result
CASTA1,070 randomizedConfirmatory global endpoint neutral
CARS208 randomizedPositive arm-motor distribution at day 90
Chinese three-arm trial84 randomized; 60 analyzedCerebrolysin better than placebo at day 21; unexplained post-randomization loss
Cochrane 2020 · no proven clinical benefit

Systematic review of randomized trials

Ziganshina LE et al. Cochrane Database of Systematic Reviews, 2020.

Seven randomized trials with 1,601 participants did not show a clear clinical benefit. All-cause mortality risk ratio was 0.90 (95% CI 0.61 to 1.32); total serious adverse events risk ratio was 1.15 (0.81 to 1.65). Nonfatal serious adverse events were more frequent with Cerebrolysin, risk ratio 2.15 (1.01 to 4.55). The trials did not supply a poolable poor-functional-outcome result.

Participants / model
1,601 participants across 7 acute ischemic stroke trials
Treatment
Cerebrolysin added to standard care versus placebo or no Cerebrolysin
Study design
Compound-specific Cochrane systematic review

The 2023 update broadened scope to similar animal-derived agents and should not be used for exact Cerebrolysin denominators.

Read the original source
CASTA · 1,070 randomized, global endpoint neutral

Randomized double-blind trial

Heiss WD et al. Stroke, 2012.

The 1,070-person trial did not show a significant benefit on its confirmatory global endpoint. A modified Rankin score of 0 to 2 occurred in 199 of 529 Cerebrolysin recipients and 208 of 541 placebo recipients.

Participants / model
1,070 people with acute ischemic stroke
Treatment
Cerebrolysin or placebo added to standard treatment
Follow-up
Acute treatment with 90-day outcome assessment
Study design
Large multicenter randomized double-blind placebo-controlled trial
Read the original source
CARS · positive smaller trial

Randomized double-blind trial

Muresanu DF et al. Stroke, 2016.

In 208 people receiving standardized rehabilitation after stroke, the Cerebrolysin arm had a better Action Research Arm Test distribution at day 90. The trial was much smaller than CASTA, and registry materials distinguish the prespecified analysis from later summaries.

Participants / model
208 people with severe arm motor impairment after acute ischemic stroke
Treatment
Cerebrolysin plus standardized rehabilitation or placebo plus rehabilitation
Follow-up
21-day treatment with 90-day assessment
Study design
Randomized double-blind placebo-controlled trial
Funding
Manufacturer involvement and author network disclosed in the publication

A positive smaller trial does not erase the neutral large confirmatory study.

Read the original source
China RCT · 84 randomized, 60 analyzed

Randomized double-blind trial

Xue LX et al. Experimental and Therapeutic Medicine, 2016.

The report says 84 people with acute ischemic stroke were randomized, but analyzes only 60 who received study intervention, 20 each with butylphthalide, Cerebrolysin, or saline placebo. At day 21, Cerebrolysin showed better NIH Stroke Scale and Barthel Index scores than placebo at reported P<0.05. Butylphthalide produced a larger NIH Stroke Scale improvement than Cerebrolysin, while their Barthel improvement did not significantly differ. The paper does not explain the 24-person randomized-to-analyzed loss, and follow-up ended at 21 days.

Participants / model
84 Chinese adults randomized within 12 hours of acute ischemic stroke; 60 analyzed, 20 per arm
Treatment
Ten days of intravenous butylphthalide, Cerebrolysin 30 mL daily, or saline placebo plus routine care
Follow-up
Ten-day treatment with assessments through day 21
Study design
Single-center randomized double-blind three-arm trial with unexplained post-randomization exclusion

The analyzed cohort is smaller than the randomized cohort.

Read the original source

Does it improve dementia?

Vascular-dementia trials show possible small score changes, but Cochrane rated the evidence very low certainty and questioned clinical importance. This is not proof of durable preservation of independence or cognition.

Cochrane dementia · very-low-certainty signals

Systematic review of randomized trials

Cui S et al. Cochrane Database of Systematic Reviews, 2019.

Six trials with 597 participants suggested small cognitive and global-response effects, but certainty was rated very low because of study limitations, inconsistency, and imprecision. The review warns that the cognitive effect may be too small to be clinically important.

Participants / model
597 participants across 6 vascular-dementia trials
Treatment
Cerebrolysin versus placebo
Study design
Cochrane systematic review
Read the original source
Glasgow review · very-low-certainty evidence

Independent systematic review

Alsulaimani RA, Quinn TJ. Cerebral Circulation, Cognition and Behavior, 2021.

The review separated animal-derived preparations and judged the Cerebrolysin evidence very low certainty. Short-term signals were not consistently maintained, and clinically meaningful functional outcomes were uncertain.

Study design
Systematic review from University of Glasgow authors
Read the original source

What is the proposed mechanism?

Laboratory and animal studies report neurotrophic, inflammatory, neurogenesis, and recovery effects, but the mixture’s active components and human exposure-response relationship are unresolved. A chromatographic fingerprint is identity control, not proof of a single active factor.

Composition study · fingerprints, no active moiety

Analytical in vitro study

Seidl LF, Aigner L. Journal of Medicine and Life, 2024.

The study compared chromatographic fingerprints and in vitro activity among porcine-brain hydrolysates using an originator reference. It does not identify one active peptide or show that market products are clinically interchangeable.

Study design
Laboratory analytical comparison
Funding
Originator material was supplied for comparison
Read the original source

What does the randomized safety record show?

The 2020 Cochrane analysis did not find a clear mortality or total-serious-adverse-event difference, but it found more nonfatal serious adverse events with Cerebrolysin. Product composition, batch comparability, hypersensitivity, interactions, pregnancy, and long-term repeated exposure remain incompletely defined.

Cochrane 2020 · no proven clinical benefit

Systematic review of randomized trials

Ziganshina LE et al. Cochrane Database of Systematic Reviews, 2020.

Seven randomized trials with 1,601 participants did not show a clear clinical benefit. All-cause mortality risk ratio was 0.90 (95% CI 0.61 to 1.32); total serious adverse events risk ratio was 1.15 (0.81 to 1.65). Nonfatal serious adverse events were more frequent with Cerebrolysin, risk ratio 2.15 (1.01 to 4.55). The trials did not supply a poolable poor-functional-outcome result.

Participants / model
1,601 participants across 7 acute ischemic stroke trials
Treatment
Cerebrolysin added to standard care versus placebo or no Cerebrolysin
Study design
Compound-specific Cochrane systematic review

The 2023 update broadened scope to similar animal-derived agents and should not be used for exact Cerebrolysin denominators.

Read the original source
Composition study · fingerprints, no active moiety

Analytical in vitro study

Seidl LF, Aigner L. Journal of Medicine and Life, 2024.

The study compared chromatographic fingerprints and in vitro activity among porcine-brain hydrolysates using an originator reference. It does not identify one active peptide or show that market products are clinically interchangeable.

Study design
Laboratory analytical comparison
Funding
Originator material was supplied for comparison
Read the original source

Where is Cerebrolysin authorized?

A CTIS record identifies a Romanian national marketing authorization and an active academic trial. The cited U.S. FDA records list no approved-drug application for Cerebrolysin. A national authorization should not be generalized into approval everywhere.

EU CTIS · active academic trial and Romanian authorization

EU clinical-trial registry record

EU CTIS 2024-515591-12-00.

The public record describes an authorized 440-person academic trial and identifies Romanian national marketing authorization 4610/2004/03 for the product used. The trial registration does not yet supply a result and the national authorization does not imply US or EU-central approval.

Participants / model
Planned 440-person stroke-recovery population
Treatment
Cerebrolysin within a randomized academic trial
Study design
Authorized prospective clinical-trial registration

Useful for current research and one specific national authorization only.

Read the original source
Drugs@FDA/openFDA · no U.S. record

Regulatory database record set

Drugs@FDA and openFDA records.

Drugs@FDA and openFDA contained no exact-name U.S. approved-drug application. This does not negate national authorization in Romania or other jurisdictions.

Study design
Exact-name U.S. approval coverage
Read the original source

Studies and sources

Cochrane 2020 · no proven clinical benefit

Systematic review of randomized trials

Ziganshina LE et al. Cochrane Database of Systematic Reviews, 2020.

Seven randomized trials with 1,601 participants did not show a clear clinical benefit. All-cause mortality risk ratio was 0.90 (95% CI 0.61 to 1.32); total serious adverse events risk ratio was 1.15 (0.81 to 1.65). Nonfatal serious adverse events were more frequent with Cerebrolysin, risk ratio 2.15 (1.01 to 4.55). The trials did not supply a poolable poor-functional-outcome result.

Participants / model
1,601 participants across 7 acute ischemic stroke trials
Treatment
Cerebrolysin added to standard care versus placebo or no Cerebrolysin
Study design
Compound-specific Cochrane systematic review

The 2023 update broadened scope to similar animal-derived agents and should not be used for exact Cerebrolysin denominators.

Read the original source
CASTA · 1,070 randomized, global endpoint neutral

Randomized double-blind trial

Heiss WD et al. Stroke, 2012.

The 1,070-person trial did not show a significant benefit on its confirmatory global endpoint. A modified Rankin score of 0 to 2 occurred in 199 of 529 Cerebrolysin recipients and 208 of 541 placebo recipients.

Participants / model
1,070 people with acute ischemic stroke
Treatment
Cerebrolysin or placebo added to standard treatment
Follow-up
Acute treatment with 90-day outcome assessment
Study design
Large multicenter randomized double-blind placebo-controlled trial
Read the original source
CARS · positive smaller trial

Randomized double-blind trial

Muresanu DF et al. Stroke, 2016.

In 208 people receiving standardized rehabilitation after stroke, the Cerebrolysin arm had a better Action Research Arm Test distribution at day 90. The trial was much smaller than CASTA, and registry materials distinguish the prespecified analysis from later summaries.

Participants / model
208 people with severe arm motor impairment after acute ischemic stroke
Treatment
Cerebrolysin plus standardized rehabilitation or placebo plus rehabilitation
Follow-up
21-day treatment with 90-day assessment
Study design
Randomized double-blind placebo-controlled trial
Funding
Manufacturer involvement and author network disclosed in the publication

A positive smaller trial does not erase the neutral large confirmatory study.

Read the original source
China RCT · 84 randomized, 60 analyzed

Randomized double-blind trial

Xue LX et al. Experimental and Therapeutic Medicine, 2016.

The report says 84 people with acute ischemic stroke were randomized, but analyzes only 60 who received study intervention, 20 each with butylphthalide, Cerebrolysin, or saline placebo. At day 21, Cerebrolysin showed better NIH Stroke Scale and Barthel Index scores than placebo at reported P<0.05. Butylphthalide produced a larger NIH Stroke Scale improvement than Cerebrolysin, while their Barthel improvement did not significantly differ. The paper does not explain the 24-person randomized-to-analyzed loss, and follow-up ended at 21 days.

Participants / model
84 Chinese adults randomized within 12 hours of acute ischemic stroke; 60 analyzed, 20 per arm
Treatment
Ten days of intravenous butylphthalide, Cerebrolysin 30 mL daily, or saline placebo plus routine care
Follow-up
Ten-day treatment with assessments through day 21
Study design
Single-center randomized double-blind three-arm trial with unexplained post-randomization exclusion

The analyzed cohort is smaller than the randomized cohort.

Read the original source
Cochrane dementia · very-low-certainty signals

Systematic review of randomized trials

Cui S et al. Cochrane Database of Systematic Reviews, 2019.

Six trials with 597 participants suggested small cognitive and global-response effects, but certainty was rated very low because of study limitations, inconsistency, and imprecision. The review warns that the cognitive effect may be too small to be clinically important.

Participants / model
597 participants across 6 vascular-dementia trials
Treatment
Cerebrolysin versus placebo
Study design
Cochrane systematic review
Read the original source
Glasgow review · very-low-certainty evidence

Independent systematic review

Alsulaimani RA, Quinn TJ. Cerebral Circulation, Cognition and Behavior, 2021.

The review separated animal-derived preparations and judged the Cerebrolysin evidence very low certainty. Short-term signals were not consistently maintained, and clinically meaningful functional outcomes were uncertain.

Study design
Systematic review from University of Glasgow authors
Read the original source
Composition study · fingerprints, no active moiety

Analytical in vitro study

Seidl LF, Aigner L. Journal of Medicine and Life, 2024.

The study compared chromatographic fingerprints and in vitro activity among porcine-brain hydrolysates using an originator reference. It does not identify one active peptide or show that market products are clinically interchangeable.

Study design
Laboratory analytical comparison
Funding
Originator material was supplied for comparison
Read the original source
EU CTIS · active academic trial and Romanian authorization

EU clinical-trial registry record

EU CTIS 2024-515591-12-00.

The public record describes an authorized 440-person academic trial and identifies Romanian national marketing authorization 4610/2004/03 for the product used. The trial registration does not yet supply a result and the national authorization does not imply US or EU-central approval.

Participants / model
Planned 440-person stroke-recovery population
Treatment
Cerebrolysin within a randomized academic trial
Study design
Authorized prospective clinical-trial registration

Useful for current research and one specific national authorization only.

Read the original source
Drugs@FDA/openFDA · no U.S. record

Regulatory database record set

Drugs@FDA and openFDA records.

Drugs@FDA and openFDA contained no exact-name U.S. approved-drug application. This does not negate national authorization in Romania or other jurisdictions.

Study design
Exact-name U.S. approval coverage
Read the original source

Why is Cerebrolysin in D tier?

D reflects inconsistent clinical results, uncertain active components, and weak certainty on patient-important outcomes. Romania has a nationally authorized product, but no US approval record was found.

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