reptides / Clomiphene

Clomiphene

Clomiphene has randomized live-birth evidence for selected female ovulatory infertility. In selected men with functional secondary hypogonadism it reliably raises LH, FSH, and testosterone. Symptom and fertility outcomes are mixed, post-AAS recovery data are weak, and healthy performance has not been tested.

Mixed-isomer selective estrogen-receptor modulator used for ovulation induction

  • US approval is for selected women with ovulatory dysfunction who desire pregnancy.
  • Selected low-testosterone men often show a large hormone response; symptom and sexual outcomes are much less certain.
  • The largest male-fertility placebo trial was negative. A newer small trial improved semen measures without measuring pregnancy or live birth.
  • Post-cycle studies mix clomiphene with natural recovery, treatment choice, hCG, testosterone, and other medicines.
  • Visual toxicity, ovarian hyperstimulation, multiple pregnancy, rising estradiol, lipid changes, and long isomer persistence matter.
Who is it for? How well does it work in PCOS? Male fertility Male low T What did China and Russia add? Post-AAS recovery Healthy performance Why can it linger? What can go wrong?

What is clomiphene FDA approved to treat?

Its US indication is selected ovulatory dysfunction in women who want pregnancy after appropriate evaluation. Male hypogonadism, male infertility, post-AAS recovery, and enhancement are off-label uses. The male evidence has to stand on its own outcomes.

US label · female ovulatory dysfunction and major warnings

FDA prescribing information

Cosette Pharmaceuticals, Inc. CLOMIPHENE CITRATE tablets. DailyMed setid 2ca373c1-4dba-4126-8616-5c533d606fe5. Updated January 31, 2025.

The US label covers ovulatory dysfunction in women desiring pregnancy, describes the mixed cis/trans isomer product, and warns about visual disorders, ovarian hyperstimulation, multiple pregnancy, liver disease, hypertriglyceridemia/pancreatitis, and prolonged isomer persistence. It says adequate controlled male-infertility efficacy evidence is absent.

Participants / model
Women with ovulatory dysfunction who desire pregnancy; label discussion also addresses unsupported male use
Treatment
Oral clomiphene citrate tablets
Follow-up
Current product record; treatment is cycle-limited in the label
Study design
Regulatory prescribing information

The label is not a male-hypogonadism or bodybuilding approval and does not provide a universal clomiphene half-life because the isomers persist differently.

Read the original source
PubChem CID 2800 · clomiphene base identity

Government substance database

National Library of Medicine. PubChem Compound Summary for CID 2800, Clomiphene.

Identifies clomiphene base as C26H28ClNO, molecular weight 406.0 g/mol, CID 2800.

Participants / model
Not applicable
Treatment
Not applicable
Follow-up
Living database record
Study design
Curated chemical identity record

The marketed citrate salt is a mixed-isomer product and has a different formula and molecular weight from the base record.

Read the original source

What do live-birth trials show for PCOS infertility?

In 626 women with PCOS, live birth was 22.5% with clomiphene, 7.2% with metformin, and 26.8% with both; adding metformin did not beat clomiphene (p=0.31). Dropout was 26.3%, 34.6%, and 23.4%, and multiple pregnancy among pregnancies was 6.0%, 0%, and 3.1%. In a later trial of 750 women, live birth was 27.5% with letrozole and 19.1% with clomiphene, an absolute difference of 8.4 percentage points (rate ratio 1.44, p=0.007). Twin pregnancy was 3.4% versus 7.4%, but that comparison was underpowered.

Use live birth, not ovulation alone
TrialClomipheneComparatorStatistical result
Clomiphene/metformin, n=62647/209 (22.5%) live birthMetformin 15/208 (7.2%); combination 56/209 (26.8%)Combination vs clomiphene p=0.31; dropout 23% to 35%
Letrozole comparison, n=75072/376 (19.1%) live birthLetrozole 103/374 (27.5%)Absolute difference 8.4 points; rate ratio 1.44; p=0.007
PCOS infertility · 626 participants and live birth

Randomized double-blind multicenter trial

Richard S. Legro, Huiman X. Barnhart, William D. Schlaff, et al.; Cooperative Multicenter Reproductive Medicine Network. New England Journal of Medicine. 2007. PMID 17287476.

Live birth was 47/209 (22.5%) with clomiphene, 15/208 (7.2%) with metformin, and 56/209 (26.8%) with both; combination versus clomiphene was p=0.31. Dropout was 26.3%, 34.6%, and 23.4%, respectively.

Participants / model
626 infertile women with polycystic ovary syndrome
Treatment
Clomiphene, extended-release metformin, or both
Follow-up
Up to 6 months, then pregnancy follow-up
Study design
Randomized double-blind multicenter comparative trial
Funding
Eunice Kennedy Shriver National Institute of Child Health and Human Development

No ultrasound follicle monitoring, hCG trigger, or intrauterine insemination was used. Multiple-pregnancy percentages use pregnancies as denominator; serious events were mostly pregnancy complications.

Read the original source
PCOS infertility · letrozole outperformed clomiphene

Randomized double-blind multicenter trial

Richard S. Legro, Robert G. Brzyski, Michael P. Diamond, et al.; NICHD Reproductive Medicine Network. New England Journal of Medicine. 2014. PMID 25006718.

Live birth was 103/374 (27.5%) with letrozole and 72/376 (19.1%) with clomiphene (rate ratio 1.44, 95% CI 1.10 to 1.87; p=0.007). Ovulation was 61.7% versus 48.3% of cycles. Twin pregnancy was 3.4% versus 7.4%, without a significant difference.

Participants / model
750 infertile women aged 18 to 40 with polycystic ovary syndrome and defined reproductive eligibility
Treatment
Letrozole versus clomiphene
Follow-up
Up to five treatment cycles with pregnancy follow-up
Study design
Randomized double-blind multicenter comparative trial
Funding
Eunice Kennedy Shriver National Institute of Child Health and Human Development

PCOS eligibility included reproductive anatomy and partner semen criteria. The study was underpowered for twins and congenital anomalies; 73.1% of infants received the planned registry physical examination.

Read the original source

Does clomiphene improve male fertility or preserve spermatogenesis?

Clomiphene maintains gonadotropin signaling and may improve semen measures in selected men. A pregnancy or live-birth benefit from treating the male partner has not been shown. The largest pregnancy-oriented placebo trial was negative. A newer small trial improved sperm concentration and motility without measuring pregnancy; a current cohort found a modest median gain and 29% of men worsened.

Male fertility: pregnancy and semen are different endpoints
StudyPopulation and designAbsolute resultLimit
WHO 1992190 couples; multicenter double-blind placebo trial; six monthsSemen unchanged; eight-month cumulative pregnancy 8.1% clomiphene vs 11.7% placeboNo benefit in this idiopathic-infertility population
Bangladesh placebo trial50 eugonadal men with idiopathic oligoasthenozoospermia randomized; 46 analyzed; 12 weeksSperm concentration 9.17→13.88 million/mL; progressive motility 14.67%→21.42%; total motile count 3.53→7.81 millionNo pregnancy or live birth; single center, short, and registered after completion
Pozzi 2026 cohort166 hypogonadal oligospermic men; retrospective; median four monthsMedian sperm concentration 4.0→5.6 million/mL; 118 improved and 48 worsenedNo control or pregnancy outcome; adverse-event discontinuations were excluded
Clomiphene plus vitamin E60 men randomized to the combination or placebo; six monthsPregnancy 11/30 vs 4/30; OR 3.76, 95% CI 1.03 to 13.64Vitamin E prevents attribution to clomiphene alone; the estimate is imprecise

Randomized sperm comparisons against testosterone gel commonly cited in this context used enclomiphene alone. Clomid contains both enclomiphene and longer-persisting zuclomiphene.

WHO male-infertility trial · no efficacy

Randomized double-blind placebo-controlled multicenter trial

World Health Organization. International Journal of Andrology. 1992. PMID 1516979.

Among 190 couples, six months of male clomiphene did not improve semen quality. Eight-month cumulative pregnancy was 8.1% with clomiphene versus 11.7% with placebo.

Participants / model
190 couples with idiopathic male semen-quality impairment and no major untreated female-factor infertility
Treatment
Oral clomiphene citrate versus placebo to male partners
Follow-up
6 months of treatment; pregnancy assessed through 8 months
Study design
Multicenter randomized double-blind placebo-controlled trial

The trial studied idiopathic male infertility, not biochemically confirmed secondary hypogonadism; pregnancy is a couple-level outcome.

Read the original source
Bangladesh placebo RCT · semen outcomes

Randomized double-blind placebo-controlled trial

Hossain MJ, et al. Clinical and Experimental Reproductive Medicine. 2025. PMID 40899280. DOI 10.5653/cerm.2024.07353.

Among 46 analyzed men, clomiphene improved sperm concentration 9.17→13.88 million/mL, progressive motility 14.67%→21.42%, total motile count 3.53→7.81 million, and testosterone 372→806 ng/dL. Nausea occurred in two and dizziness in three.

Participants / model
50 eugonadal men with idiopathic oligoasthenozoospermia randomized; 46 analyzed
Treatment
Clomiphene citrate versus placebo
Follow-up
12 weeks
Study design
Single-center randomized double-blind placebo-controlled trial

No pregnancy or live-birth endpoint. The trial was registered after completion; funding was not stated and no relevant conflict was reported.

Read the original source
Pozzi et al. · 166-man sperm-response cohort

Retrospective cohort

Pozzi E, De Luca S, Birolini G, et al. World Journal of Men's Health. 2026. PMID 42533482. DOI 10.5534/wjmh.250371.

151/166 reached testosterone ≥3.5 ng/mL. Median sperm concentration rose 4.0→5.6 million/mL; 118 improved and 48 worsened by a median 3.3 million/mL.

Participants / model
166 hypogonadal oligospermic men
Treatment
Clomiphene citrate
Follow-up
At least 3 months; median follow-up 4 months
Study design
Single-center retrospective cohort

No comparator or pregnancy outcome, 11% dropout, exclusion of adverse-event discontinuations, and a white-European cohort limit inference. The authors reported no disclosure.

Read the original source
Ghanem et al. · clomiphene plus vitamin E

Randomized placebo-controlled combination trial

Ghanem H, Shaeer O, El-Segini A. Fertility and Sterility. 2010;93(7):2232-2235. PMID 19268928.

Pregnancy occurred in 11/30 couples assigned clomiphene plus vitamin E and 4/30 assigned placebo; OR 3.76 (95% CI 1.03 to 13.64).

Participants / model
60 men with idiopathic infertility and their partners
Treatment
Clomiphene plus vitamin E versus placebo
Follow-up
6 months
Study design
Randomized controlled combination-treatment trial

Vitamin E prevents attribution to clomiphene alone, and the confidence interval is wide.

Read the original source

How strong is the evidence for low testosterone and symptoms in men?

The hormone effect is repeatable in selected men with a responsive pituitary and testes. In the best placebo trial, mean testosterone rose from about 226 to 688 ng/dL over 12 weeks while placebo stayed near 220. The same trial found no between-group improvement in its aggregate symptom score or most sexual complaints, no fat loss or endothelial benefit, and an HDL fall. Uncontrolled cohorts often report symptom improvement, but blinded evidence remains mixed.

Hormone response, symptoms, and durability
EvidenceHormone resultSymptoms or durabilityLimit
Soares placebo RCTTotal testosterone about 225.5→687.9 ng/dL over 12 weeksNo between-group aggregate symptom or most sexual-complaint benefit; lean mass +2.2 kg; HDL −8.5 mg/dL67/78 analyzed; obese symptomatic men with T ≤300; short and single center
Habous active-comparator RCTTestosterone rose in clomiphene, hCG, and combination groupsqADAM improved in all armsNo placebo; abstract reports n=282 while group counts total 283
Krzastek long-term cohortAmong 120 men treated beyond three years, 88% were eugonadal77% reported symptom improvement; 8% reported side effectsRetrospective study of selected long-term continuers; no comparator
Huijben cohortMean testosterone 9→16 nmol/L; it fell after 48/52 withdrawal trials74% reported improvement; adverse-event documentation was absent in 130/153 chartsHeterogeneous retrospective cohort with loss, stopping, and switching
Kim 2026 cohort136/292 (47%) met ≥400 ng/dL plus a ≥200-ng/dL riseNo symptom outcomeShort retrospective assessment; higher LH and prior androgen deprivation predicted failure
78 men · hormones and body-composition surrogates

Randomized double-blind placebo-controlled trial

Andressa Heimbecher Soares, Nidia Celeste Horie, Lucas Augusto Piccinin Chiang, et al. International Journal of Obesity. 2018. PMID 29777228.

Seventy-eight men were randomized and 67 analyzed at 12 weeks. Hormones and several lean-mass measures rose; BMI, waist, fat mass, endothelial function, and most sexual complaints were unchanged, and HDL fell. No clomiphene participant discontinued for an adverse event.

Participants / model
78 men with obesity-associated secondary hypogonadism randomized; 67 analyzed at 12 weeks
Treatment
Oral clomiphene citrate versus placebo
Follow-up
12 weeks
Study design
Single-center randomized double-blind placebo-controlled trial

Short single-center surrogate trial without a testosterone-replacement comparator, fertility endpoints, long-term symptoms, or cardiovascular outcomes; diet and activity were not standardized.

Read the original source
Habous et al. · clomiphene vs hCG vs combination

Randomized active-comparator trial

Habous M, Giona S, Tealab A, et al. BJU International. 2018;122(5):889-897. PMID 29772111. DOI 10.1111/bju.14401.

The abstract reports testosterone and qADAM improvement in clomiphene, hCG, and combination arms, with the largest qADAM gain in the combination arm.

Participants / model
Men with hypogonadism; abstract reports total n=282 while listed group counts sum to 283
Treatment
Clomiphene, hCG, or both
Follow-up
3 months
Study design
Randomized active-comparator study without placebo

No semen or pregnancy endpoint. The abstract does not resolve the adverse-event, funding, or denominator details.

Read the original source
Krzastek et al. · 400-man retrospective cohort

Retrospective two-center cohort

Krzastek SC, Sharma D, Abdullah N, et al. Journal of Urology. 2019;202(5):1029-1035. PMID 31216250. DOI 10.1097/JU.0000000000000396.

Of 400 treated men, 120 remained treated beyond three years; in that selected group 88% were eugonadal, 77% reported symptom improvement, and 8% reported side effects.

Participants / model
400 men treated for hypogonadism; 120 treated longer than three years
Treatment
Clomiphene citrate
Follow-up
Mean 25.5 months; selected subgroup beyond 3 years
Study design
Retrospective two-center cohort

No untreated control and strong survivor or continuation selection.

Read the original source
Huijben et al. · response, withdrawal, and chart gaps

Retrospective cohort

Huijben M, Huijsmans RLN, Lock MTWT, de Kemp VF, de Kort LMO, van Breda JHMK. Endocrinology, Diabetes & Metabolism. 2023;6:e416. PMID 36998229.

Mean testosterone rose 9→16 nmol/L and 74% reported improvement. Testosterone fell after 48/52 withdrawal trials. Recorded adverse events occurred in 16/153, but adverse-event documentation was absent in 130 charts.

Participants / model
153 heterogeneous men treated for hypogonadism
Treatment
Clomiphene citrate
Follow-up
Retrospective follow-up with variable duration and withdrawal trials
Study design
Single-center retrospective cohort

No validated symptom tool or control. At endpoint only 43 remained followed; 26 were lost, 71 stopped, and 14 switched to testosterone. Authors reported no funding or conflicts.

Read the original source
Kim et al. · stricter biochemical response cohort

Retrospective response-predictor cohort

Kim JK, et al. Journal of Sexual Medicine. 2026. PMID 42251758. DOI 10.1093/jsxmed/qdag159.

136/292 men (47%) reached testosterone ≥400 ng/dL plus a ≥200-ng/dL rise within 12 weeks. Higher baseline LH predicted lower response odds, and prior androgen-deprivation therapy had OR 0.11.

Participants / model
292 men with low or borderline testosterone plus symptoms or objective signs
Treatment
Clomiphene citrate
Follow-up
Response assessed within 12 weeks
Study design
Retrospective clinical cohort
Funding
NIH/NCI core support listed; no declared conflict

No symptom outcomes and short follow-up; the response definition is stricter than simple normalization.

Read the original source

Why do the local studies not overturn the larger trials?

The Russian report described 6 conceptions among 30 men receiving clomiphene. Treatment was not randomized and untreated controls chose observation. The Bangladesh placebo trial improved semen measures but measured no pregnancy. A Chinese abstract in women used the same herbal co-treatment in both arms and favored letrozole for ovulation and pregnancy without measuring live birth. The WHO male-pregnancy result remained negative.

Russian report · nonrandomized male-infertility comparison

Russian prospective clinical comparative study

N. S. Kravtsova, R. V. Rozhivanov, and D. G. Kurbatov. Проблемы эндокринологии. 2016;62(2):37 to 41. DOI 10.14341/probl201662237-41.

The report describes 80 men: clomiphene 30, hCG 10, hCG plus recombinant FSH 30, and self-selected no-treatment control 10. At six months, conception was 6/30 in the clomiphene group and oligo-teratozoospermia reportedly resolved in 19/30; three deteriorated.

Participants / model
80 men with pathospermia and infertility; treatment selection and control participation were not randomized
Treatment
Clomiphene, hCG, hCG plus recombinant FSH, or observation
Follow-up
3 months with continuation to 6 months
Study design
Prospective comparative study with stratification among treated groups and self-selected untreated controls

There was no randomized placebo comparison, controls self-selected, partner factors confound conception, treatment groups differed, and the study was not powered for safety.

Read the original source
Bangladesh placebo RCT · semen outcomes

Randomized double-blind placebo-controlled trial

Hossain MJ, et al. Clinical and Experimental Reproductive Medicine. 2025. PMID 40899280. DOI 10.5653/cerm.2024.07353.

Among 46 analyzed men, clomiphene improved sperm concentration 9.17→13.88 million/mL, progressive motility 14.67%→21.42%, total motile count 3.53→7.81 million, and testosterone 372→806 ng/dL. Nausea occurred in two and dizziness in three.

Participants / model
50 eugonadal men with idiopathic oligoasthenozoospermia randomized; 46 analyzed
Treatment
Clomiphene citrate versus placebo
Follow-up
12 weeks
Study design
Single-center randomized double-blind placebo-controlled trial

No pregnancy or live-birth endpoint. The trial was registered after completion; funding was not stated and no relevant conflict was reported.

Read the original source
Chinese abstract · clomiphene versus letrozole with co-treatment

Chinese randomized comparative clinical study

王鑫, 张丛轶, 王静, 李静, 李娅. 转化医学杂志. 2025;14:156 to 160.

The native and publisher-translated abstracts report 206 women randomized 103 per group. Both groups received compound Xuanju capsules; letrozole versus clomiphene had higher reported ovulation (72.82% versus 59.22%) and pregnancy (45.63% versus 31.07%) over three cycles.

Participants / model
206 women with ovulatory-disorder infertility
Treatment
Compound Xuanju plus clomiphene versus compound Xuanju plus letrozole
Follow-up
Three treatment cycles
Study design
Randomized-number-table comparative study reported in abstract

Shared herbal co-treatment, unclear blinding, no live-birth endpoint, and abstract-only reporting limit inference.

Read the original source
WHO male-infertility trial · no efficacy

Randomized double-blind placebo-controlled multicenter trial

World Health Organization. International Journal of Andrology. 1992. PMID 1516979.

Among 190 couples, six months of male clomiphene did not improve semen quality. Eight-month cumulative pregnancy was 8.1% with clomiphene versus 11.7% with placebo.

Participants / model
190 couples with idiopathic male semen-quality impairment and no major untreated female-factor infertility
Treatment
Oral clomiphene citrate versus placebo to male partners
Follow-up
6 months of treatment; pregnancy assessed through 8 months
Study design
Multicenter randomized double-blind placebo-controlled trial

The trial studied idiopathic male infertility, not biochemically confirmed secondary hypogonadism; pregnancy is a couple-level outcome.

Read the original source
PCOS infertility · letrozole outperformed clomiphene

Randomized double-blind multicenter trial

Richard S. Legro, Robert G. Brzyski, Michael P. Diamond, et al.; NICHD Reproductive Medicine Network. New England Journal of Medicine. 2014. PMID 25006718.

Live birth was 103/374 (27.5%) with letrozole and 72/376 (19.1%) with clomiphene (rate ratio 1.44, 95% CI 1.10 to 1.87; p=0.007). Ovulation was 61.7% versus 48.3% of cycles. Twin pregnancy was 3.4% versus 7.4%, without a significant difference.

Participants / model
750 infertile women aged 18 to 40 with polycystic ovary syndrome and defined reproductive eligibility
Treatment
Letrozole versus clomiphene
Follow-up
Up to five treatment cycles with pregnancy follow-up
Study design
Randomized double-blind multicenter comparative trial
Funding
Eunice Kennedy Shriver National Institute of Child Health and Human Development

PCOS eligibility included reproductive anatomy and partner semen criteria. The study was underpowered for twins and congenital anomalies; 73.1% of infants received the planned registry physical examination.

Read the original source

Does clomiphene make post-cycle therapy proven?

Three clinical reports suggest earlier hormone or semen recovery during clomiphene-containing care, but none isolates clomiphene. Natural recovery, treatment choice, hCG, short testosterone bridging, aromatase inhibitors, FSH, different AAS histories, and clinical follow-up all affect the result.

What the post-AAS studies measured
StudyDesignResultLimit
Al Hashimi 2022520 AAS users observed for three months; 463 then chose individualized treatment and 57 observationTreated men recovered hormones, IIEF, testicular size, and semen faster; 14 pregnancies among 94 infertility presentations by month 12The paper calls the study randomized, but groups followed patient choice; treatment also used hCG, tamoxifen, aromatase inhibitor, or FSH
Henriksen 2024 pilot81 screened, 17 eligible, 10 completed; all received clomiphene, six had a testosterone bridge, seven received indicated hCGFive of 10 reached or ended within the normal testosterone range; no serious adverse eventOpen feasibility study; symptoms did not track testosterone response; heavy selection and mixed treatment
İbis 2025/2026 cohort79 short-term AAS users managed with observation, clomiphene, or clomiphene plus hCGAll groups normalized hormones by month 6; 12-month normozoospermia 69.2%, 87.5%, and 58.6%Retrospective and nonrandomized; no pregnancy or live-birth endpoint

These studies describe supervised research care. They do not define a self-directed protocol.

Al Hashimi et al. · chosen mixed-treatment AAS cohort

Prospective nonrandomized comparative cohort

Al Hashimi M, et al. Andrologia. 2022. PMID 36065528. DOI 10.1111/and.14576.

After three months of observation, 463 of 520 former AAS users chose individualized treatment and 57 continued observation. Treated men recovered hormones, sexual function, testicular size, and semen earlier; 14 pregnancies were reported among 94 infertility presentations by month 12.

Participants / model
520 men after anabolic-androgenic steroid use
Treatment
Individualized hCG plus clomiphene, sometimes with tamoxifen, aromatase inhibitor, or FSH, versus observation
Follow-up
Up to 12 months after an initial 3-month observation period
Study design
Prospective cohort assigned by patient choice despite the paper's randomized label

No clomiphene-only arm. Baseline and treatment-selection confounding are severe. The paper inconsistently reports 74 versus 94 infertility cases. The authors reported no conflicts.

Read the original source
Henriksen et al. · mixed-intervention pilot

Open uncontrolled feasibility pilot

Henriksen HCB, et al. Performance Enhancement & Health. 2024;12(3):100283. DOI 10.1016/j.peh.2024.100283.

Of 81 screened and 17 eligible men, 10 completed. Five reached or ended within the normal testosterone range; withdrawal symptoms did not track testosterone response. Seven reported some clomiphene adverse effect at week 4, falling to three at week 16; no serious adverse event.

Participants / model
Men with long-term AAS use in substance-use-disorder care; 10 completers
Treatment
Clomiphene for all; six also received a short testosterone bridge and seven indicated hCG
Follow-up
16 weeks
Study design
Open uncontrolled feasibility pilot with mixed interventions
Funding
Public Norwegian and Oslo University Hospital support

Severe screening selection, co-treatment, clinical care, and time prevent clomiphene-only attribution.

Read the original source
İbis et al. · nonrandomized PCT cohort

Retrospective dual-center comparative cohort

İbis MA, et al. BJU International. Epub 2025. PMID 41147237. DOI 10.1111/bju.70059.

In 79 men, clomiphene-containing groups recovered hormones and semen earlier. All groups normalized hormones by month 6; at month 12 normozoospermia was 69.2% clomiphene, 87.5% clomiphene plus hCG, and 58.6% untreated.

Participants / model
79 recreational bodybuilders after no more than 6 months of AAS use with documented normal pre-cycle hormones and semen
Treatment
Observation, clomiphene, or clomiphene plus hCG; FSH suggested for five men
Follow-up
12 months
Study design
Retrospective nonrandomized dual-center cohort

Natural recovery was substantial, treatment was not randomized, adjusted estimates were imprecise, and there was no pregnancy or live-birth endpoint. Adverse-event and funding details remain unresolved.

Read the original source

Does clomiphene improve muscle or performance in healthy men?

No controlled trial in the cited evidence measured hypertrophy, maximal strength, power, endurance, training adaptation, or recovery in healthy eugonadal athletes. The 2.2 kg lean-mass increase came from obese symptomatic men with low testosterone and lasted 12 weeks. It did not establish better performance.

Enclomiphene is the isolated trans isomer. Clomid is a mixture of enclomiphene and zuclomiphene, so enclomiphene-only trials need their own label.

78 men · hormones and body-composition surrogates

Randomized double-blind placebo-controlled trial

Andressa Heimbecher Soares, Nidia Celeste Horie, Lucas Augusto Piccinin Chiang, et al. International Journal of Obesity. 2018. PMID 29777228.

Seventy-eight men were randomized and 67 analyzed at 12 weeks. Hormones and several lean-mass measures rose; BMI, waist, fat mass, endothelial function, and most sexual complaints were unchanged, and HDL fell. No clomiphene participant discontinued for an adverse event.

Participants / model
78 men with obesity-associated secondary hypogonadism randomized; 67 analyzed at 12 weeks
Treatment
Oral clomiphene citrate versus placebo
Follow-up
12 weeks
Study design
Single-center randomized double-blind placebo-controlled trial

Short single-center surrogate trial without a testosterone-replacement comparator, fertility endpoints, long-term symptoms, or cardiovascular outcomes; diet and activity were not standardized.

Read the original source
US label · female ovulatory dysfunction and major warnings

FDA prescribing information

Cosette Pharmaceuticals, Inc. CLOMIPHENE CITRATE tablets. DailyMed setid 2ca373c1-4dba-4126-8616-5c533d606fe5. Updated January 31, 2025.

The US label covers ovulatory dysfunction in women desiring pregnancy, describes the mixed cis/trans isomer product, and warns about visual disorders, ovarian hyperstimulation, multiple pregnancy, liver disease, hypertriglyceridemia/pancreatitis, and prolonged isomer persistence. It says adequate controlled male-infertility efficacy evidence is absent.

Participants / model
Women with ovulatory dysfunction who desire pregnancy; label discussion also addresses unsupported male use
Treatment
Oral clomiphene citrate tablets
Follow-up
Current product record; treatment is cycle-limited in the label
Study design
Regulatory prescribing information

The label is not a male-hypogonadism or bodybuilding approval and does not provide a universal clomiphene half-life because the isomers persist differently.

Read the original source

Does clomiphene have one reliable half-life?

Clomiphene is an isomer mixture, and the cis isomer zuclomiphene persists much longer than the trans isomer. The label reports prolonged radiolabeled material and detectable zuclomiphene beyond a month, so one parent-drug half-life would be misleading.

US label · female ovulatory dysfunction and major warnings

FDA prescribing information

Cosette Pharmaceuticals, Inc. CLOMIPHENE CITRATE tablets. DailyMed setid 2ca373c1-4dba-4126-8616-5c533d606fe5. Updated January 31, 2025.

The US label covers ovulatory dysfunction in women desiring pregnancy, describes the mixed cis/trans isomer product, and warns about visual disorders, ovarian hyperstimulation, multiple pregnancy, liver disease, hypertriglyceridemia/pancreatitis, and prolonged isomer persistence. It says adequate controlled male-infertility efficacy evidence is absent.

Participants / model
Women with ovulatory dysfunction who desire pregnancy; label discussion also addresses unsupported male use
Treatment
Oral clomiphene citrate tablets
Follow-up
Current product record; treatment is cycle-limited in the label
Study design
Regulatory prescribing information

The label is not a male-hypogonadism or bodybuilding approval and does not provide a universal clomiphene half-life because the isomers persist differently.

Read the original source

Which warnings matter before anyone calls it a harmless SERM?

The label warns about visual injury, ovarian hyperstimulation, multiple pregnancy, liver disease, high triglycerides, pancreatitis, and thrombotic events. Male studies report rising estradiol, breast tenderness, mood change, blurred vision, dizziness, fatigue, headache, and gastrointestinal symptoms. Most cohorts are too short or too selected to estimate uncommon or long-term harm.

The 400-man series' 8% side-effect figure came from 120 men who remained treated beyond three years. In Huijben, adverse-event documentation was missing in 130 of 153 charts.

A VA database study matched 2,518 clomiphene users to 2,518 testosterone users and found fewer coded events with clomiphene. Infertility remained coded in 895 versus 41, while smoking, severity, symptoms, free testosterone, bone density, and medication differences were unresolved. Mortality was 1.83% versus 10.13%; the design cannot make that a treatment effect.

US label · female ovulatory dysfunction and major warnings

FDA prescribing information

Cosette Pharmaceuticals, Inc. CLOMIPHENE CITRATE tablets. DailyMed setid 2ca373c1-4dba-4126-8616-5c533d606fe5. Updated January 31, 2025.

The US label covers ovulatory dysfunction in women desiring pregnancy, describes the mixed cis/trans isomer product, and warns about visual disorders, ovarian hyperstimulation, multiple pregnancy, liver disease, hypertriglyceridemia/pancreatitis, and prolonged isomer persistence. It says adequate controlled male-infertility efficacy evidence is absent.

Participants / model
Women with ovulatory dysfunction who desire pregnancy; label discussion also addresses unsupported male use
Treatment
Oral clomiphene citrate tablets
Follow-up
Current product record; treatment is cycle-limited in the label
Study design
Regulatory prescribing information

The label is not a male-hypogonadism or bodybuilding approval and does not provide a universal clomiphene half-life because the isomers persist differently.

Read the original source
Krzastek et al. · 400-man retrospective cohort

Retrospective two-center cohort

Krzastek SC, Sharma D, Abdullah N, et al. Journal of Urology. 2019;202(5):1029-1035. PMID 31216250. DOI 10.1097/JU.0000000000000396.

Of 400 treated men, 120 remained treated beyond three years; in that selected group 88% were eugonadal, 77% reported symptom improvement, and 8% reported side effects.

Participants / model
400 men treated for hypogonadism; 120 treated longer than three years
Treatment
Clomiphene citrate
Follow-up
Mean 25.5 months; selected subgroup beyond 3 years
Study design
Retrospective two-center cohort

No untreated control and strong survivor or continuation selection.

Read the original source
Huijben et al. · response, withdrawal, and chart gaps

Retrospective cohort

Huijben M, Huijsmans RLN, Lock MTWT, de Kemp VF, de Kort LMO, van Breda JHMK. Endocrinology, Diabetes & Metabolism. 2023;6:e416. PMID 36998229.

Mean testosterone rose 9→16 nmol/L and 74% reported improvement. Testosterone fell after 48/52 withdrawal trials. Recorded adverse events occurred in 16/153, but adverse-event documentation was absent in 130 charts.

Participants / model
153 heterogeneous men treated for hypogonadism
Treatment
Clomiphene citrate
Follow-up
Retrospective follow-up with variable duration and withdrawal trials
Study design
Single-center retrospective cohort

No validated symptom tool or control. At endpoint only 43 remained followed; 26 were lost, 71 stopped, and 14 switched to testosterone. Authors reported no funding or conflicts.

Read the original source
VA cohort · comparative associations

Matched retrospective database cohort

Testosterone Versus Clomiphene Treatment of Hypogonadism: A Retrospective Analysis in US Veterans. Andrology. 2026. PMID 42015850. DOI 10.1111/andr.70229.

2,518 clomiphene users were matched to 2,518 testosterone users. Coded cardiovascular, polycythemia, osteoporosis, and mortality outcomes were lower with clomiphene; mortality was 1.83% versus 10.13%.

Participants / model
5,036 matched US veterans treated for hypogonadism
Treatment
Clomiphene citrate versus testosterone
Follow-up
Mean follow-up about 3.4 to 3.8 years
Study design
Retrospective administrative-database comparison

Infertility remained profoundly imbalanced (895 vs 41), and smoking, severity, medicines, symptoms, free testosterone, and bone density were omitted. The mortality contrast is not causal. Authors reported no funding or conflicts.

Read the original source
78 men · hormones and body-composition surrogates

Randomized double-blind placebo-controlled trial

Andressa Heimbecher Soares, Nidia Celeste Horie, Lucas Augusto Piccinin Chiang, et al. International Journal of Obesity. 2018. PMID 29777228.

Seventy-eight men were randomized and 67 analyzed at 12 weeks. Hormones and several lean-mass measures rose; BMI, waist, fat mass, endothelial function, and most sexual complaints were unchanged, and HDL fell. No clomiphene participant discontinued for an adverse event.

Participants / model
78 men with obesity-associated secondary hypogonadism randomized; 67 analyzed at 12 weeks
Treatment
Oral clomiphene citrate versus placebo
Follow-up
12 weeks
Study design
Single-center randomized double-blind placebo-controlled trial

Short single-center surrogate trial without a testosterone-replacement comparator, fertility endpoints, long-term symptoms, or cardiovascular outcomes; diet and activity were not standardized.

Read the original source

Studies and sources

US label · female ovulatory dysfunction and major warnings

FDA prescribing information

Cosette Pharmaceuticals, Inc. CLOMIPHENE CITRATE tablets. DailyMed setid 2ca373c1-4dba-4126-8616-5c533d606fe5. Updated January 31, 2025.

The US label covers ovulatory dysfunction in women desiring pregnancy, describes the mixed cis/trans isomer product, and warns about visual disorders, ovarian hyperstimulation, multiple pregnancy, liver disease, hypertriglyceridemia/pancreatitis, and prolonged isomer persistence. It says adequate controlled male-infertility efficacy evidence is absent.

Participants / model
Women with ovulatory dysfunction who desire pregnancy; label discussion also addresses unsupported male use
Treatment
Oral clomiphene citrate tablets
Follow-up
Current product record; treatment is cycle-limited in the label
Study design
Regulatory prescribing information

The label is not a male-hypogonadism or bodybuilding approval and does not provide a universal clomiphene half-life because the isomers persist differently.

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PCOS infertility · 626 participants and live birth

Randomized double-blind multicenter trial

Richard S. Legro, Huiman X. Barnhart, William D. Schlaff, et al.; Cooperative Multicenter Reproductive Medicine Network. New England Journal of Medicine. 2007. PMID 17287476.

Live birth was 47/209 (22.5%) with clomiphene, 15/208 (7.2%) with metformin, and 56/209 (26.8%) with both; combination versus clomiphene was p=0.31. Dropout was 26.3%, 34.6%, and 23.4%, respectively.

Participants / model
626 infertile women with polycystic ovary syndrome
Treatment
Clomiphene, extended-release metformin, or both
Follow-up
Up to 6 months, then pregnancy follow-up
Study design
Randomized double-blind multicenter comparative trial
Funding
Eunice Kennedy Shriver National Institute of Child Health and Human Development

No ultrasound follicle monitoring, hCG trigger, or intrauterine insemination was used. Multiple-pregnancy percentages use pregnancies as denominator; serious events were mostly pregnancy complications.

Read the original source
PCOS infertility · letrozole outperformed clomiphene

Randomized double-blind multicenter trial

Richard S. Legro, Robert G. Brzyski, Michael P. Diamond, et al.; NICHD Reproductive Medicine Network. New England Journal of Medicine. 2014. PMID 25006718.

Live birth was 103/374 (27.5%) with letrozole and 72/376 (19.1%) with clomiphene (rate ratio 1.44, 95% CI 1.10 to 1.87; p=0.007). Ovulation was 61.7% versus 48.3% of cycles. Twin pregnancy was 3.4% versus 7.4%, without a significant difference.

Participants / model
750 infertile women aged 18 to 40 with polycystic ovary syndrome and defined reproductive eligibility
Treatment
Letrozole versus clomiphene
Follow-up
Up to five treatment cycles with pregnancy follow-up
Study design
Randomized double-blind multicenter comparative trial
Funding
Eunice Kennedy Shriver National Institute of Child Health and Human Development

PCOS eligibility included reproductive anatomy and partner semen criteria. The study was underpowered for twins and congenital anomalies; 73.1% of infants received the planned registry physical examination.

Read the original source
WHO male-infertility trial · no efficacy

Randomized double-blind placebo-controlled multicenter trial

World Health Organization. International Journal of Andrology. 1992. PMID 1516979.

Among 190 couples, six months of male clomiphene did not improve semen quality. Eight-month cumulative pregnancy was 8.1% with clomiphene versus 11.7% with placebo.

Participants / model
190 couples with idiopathic male semen-quality impairment and no major untreated female-factor infertility
Treatment
Oral clomiphene citrate versus placebo to male partners
Follow-up
6 months of treatment; pregnancy assessed through 8 months
Study design
Multicenter randomized double-blind placebo-controlled trial

The trial studied idiopathic male infertility, not biochemically confirmed secondary hypogonadism; pregnancy is a couple-level outcome.

Read the original source
78 men · hormones and body-composition surrogates

Randomized double-blind placebo-controlled trial

Andressa Heimbecher Soares, Nidia Celeste Horie, Lucas Augusto Piccinin Chiang, et al. International Journal of Obesity. 2018. PMID 29777228.

Seventy-eight men were randomized and 67 analyzed at 12 weeks. Hormones and several lean-mass measures rose; BMI, waist, fat mass, endothelial function, and most sexual complaints were unchanged, and HDL fell. No clomiphene participant discontinued for an adverse event.

Participants / model
78 men with obesity-associated secondary hypogonadism randomized; 67 analyzed at 12 weeks
Treatment
Oral clomiphene citrate versus placebo
Follow-up
12 weeks
Study design
Single-center randomized double-blind placebo-controlled trial

Short single-center surrogate trial without a testosterone-replacement comparator, fertility endpoints, long-term symptoms, or cardiovascular outcomes; diet and activity were not standardized.

Read the original source
Russian report · nonrandomized male-infertility comparison

Russian prospective clinical comparative study

N. S. Kravtsova, R. V. Rozhivanov, and D. G. Kurbatov. Проблемы эндокринологии. 2016;62(2):37 to 41. DOI 10.14341/probl201662237-41.

The report describes 80 men: clomiphene 30, hCG 10, hCG plus recombinant FSH 30, and self-selected no-treatment control 10. At six months, conception was 6/30 in the clomiphene group and oligo-teratozoospermia reportedly resolved in 19/30; three deteriorated.

Participants / model
80 men with pathospermia and infertility; treatment selection and control participation were not randomized
Treatment
Clomiphene, hCG, hCG plus recombinant FSH, or observation
Follow-up
3 months with continuation to 6 months
Study design
Prospective comparative study with stratification among treated groups and self-selected untreated controls

There was no randomized placebo comparison, controls self-selected, partner factors confound conception, treatment groups differed, and the study was not powered for safety.

Read the original source
Chinese abstract · clomiphene versus letrozole with co-treatment

Chinese randomized comparative clinical study

王鑫, 张丛轶, 王静, 李静, 李娅. 转化医学杂志. 2025;14:156 to 160.

The native and publisher-translated abstracts report 206 women randomized 103 per group. Both groups received compound Xuanju capsules; letrozole versus clomiphene had higher reported ovulation (72.82% versus 59.22%) and pregnancy (45.63% versus 31.07%) over three cycles.

Participants / model
206 women with ovulatory-disorder infertility
Treatment
Compound Xuanju plus clomiphene versus compound Xuanju plus letrozole
Follow-up
Three treatment cycles
Study design
Randomized-number-table comparative study reported in abstract

Shared herbal co-treatment, unclear blinding, no live-birth endpoint, and abstract-only reporting limit inference.

Read the original source
PubChem CID 2800 · clomiphene base identity

Government substance database

National Library of Medicine. PubChem Compound Summary for CID 2800, Clomiphene.

Identifies clomiphene base as C26H28ClNO, molecular weight 406.0 g/mol, CID 2800.

Participants / model
Not applicable
Treatment
Not applicable
Follow-up
Living database record
Study design
Curated chemical identity record

The marketed citrate salt is a mixed-isomer product and has a different formula and molecular weight from the base record.

Read the original source
Dadhich et al. · chosen-treatment symptom cohort

Prospective nonrandomized comparative cohort

Dadhich P, Ramasamy R, Scovell J, Wilken N, Lipshultz L. Indian Journal of Urology. 2017;33(3):236-240. PMID 28717276. DOI 10.4103/iju.IJU_372_16.

Among 23 men choosing clomiphene, testosterone rose 235→438 ng/dL and overall ADAM/qADAM scores improved, while the libido item worsened 3.75→3.2 (p=.04).

Participants / model
75 symptomatic men; 23 chose clomiphene and 52 chose testosterone
Treatment
Patient-chosen clomiphene or testosterone therapy
Follow-up
Prospective follow-up; duration differed between groups
Study design
Nonrandomized prospective comparative cohort

Clomiphene users were younger and fertility-motivated; treatment choice and unequal follow-up confound comparison. The authors reported no funding or conflicts.

Read the original source
Habous et al. · clomiphene vs hCG vs combination

Randomized active-comparator trial

Habous M, Giona S, Tealab A, et al. BJU International. 2018;122(5):889-897. PMID 29772111. DOI 10.1111/bju.14401.

The abstract reports testosterone and qADAM improvement in clomiphene, hCG, and combination arms, with the largest qADAM gain in the combination arm.

Participants / model
Men with hypogonadism; abstract reports total n=282 while listed group counts sum to 283
Treatment
Clomiphene, hCG, or both
Follow-up
3 months
Study design
Randomized active-comparator study without placebo

No semen or pregnancy endpoint. The abstract does not resolve the adverse-event, funding, or denominator details.

Read the original source
Krzastek et al. · 400-man retrospective cohort

Retrospective two-center cohort

Krzastek SC, Sharma D, Abdullah N, et al. Journal of Urology. 2019;202(5):1029-1035. PMID 31216250. DOI 10.1097/JU.0000000000000396.

Of 400 treated men, 120 remained treated beyond three years; in that selected group 88% were eugonadal, 77% reported symptom improvement, and 8% reported side effects.

Participants / model
400 men treated for hypogonadism; 120 treated longer than three years
Treatment
Clomiphene citrate
Follow-up
Mean 25.5 months; selected subgroup beyond 3 years
Study design
Retrospective two-center cohort

No untreated control and strong survivor or continuation selection.

Read the original source
Huijben et al. · response, withdrawal, and chart gaps

Retrospective cohort

Huijben M, Huijsmans RLN, Lock MTWT, de Kemp VF, de Kort LMO, van Breda JHMK. Endocrinology, Diabetes & Metabolism. 2023;6:e416. PMID 36998229.

Mean testosterone rose 9→16 nmol/L and 74% reported improvement. Testosterone fell after 48/52 withdrawal trials. Recorded adverse events occurred in 16/153, but adverse-event documentation was absent in 130 charts.

Participants / model
153 heterogeneous men treated for hypogonadism
Treatment
Clomiphene citrate
Follow-up
Retrospective follow-up with variable duration and withdrawal trials
Study design
Single-center retrospective cohort

No validated symptom tool or control. At endpoint only 43 remained followed; 26 were lost, 71 stopped, and 14 switched to testosterone. Authors reported no funding or conflicts.

Read the original source
Anno et al. · one-year AMS cohort

Retrospective cohort

Anno Y, et al. International Journal of Urology. 2026. PMID 41250569. DOI 10.1111/iju.70289.

In 54 symptomatic Japanese men, testosterone and total Aging Males' Symptoms score improved over one year, while the sexual-dysfunction domain did not.

Participants / model
54 Japanese men with late-onset hypogonadism symptoms
Treatment
Clomiphene citrate
Follow-up
1 year
Study design
Retrospective uncontrolled cohort
Funding
PubMed record lists no grants; authors reported no conflict

The abstract does not report absolute outcome values or full adverse-event detail.

Read the original source
Kim et al. · stricter biochemical response cohort

Retrospective response-predictor cohort

Kim JK, et al. Journal of Sexual Medicine. 2026. PMID 42251758. DOI 10.1093/jsxmed/qdag159.

136/292 men (47%) reached testosterone ≥400 ng/dL plus a ≥200-ng/dL rise within 12 weeks. Higher baseline LH predicted lower response odds, and prior androgen-deprivation therapy had OR 0.11.

Participants / model
292 men with low or borderline testosterone plus symptoms or objective signs
Treatment
Clomiphene citrate
Follow-up
Response assessed within 12 weeks
Study design
Retrospective clinical cohort
Funding
NIH/NCI core support listed; no declared conflict

No symptom outcomes and short follow-up; the response definition is stricter than simple normalization.

Read the original source
VA cohort · comparative associations

Matched retrospective database cohort

Testosterone Versus Clomiphene Treatment of Hypogonadism: A Retrospective Analysis in US Veterans. Andrology. 2026. PMID 42015850. DOI 10.1111/andr.70229.

2,518 clomiphene users were matched to 2,518 testosterone users. Coded cardiovascular, polycythemia, osteoporosis, and mortality outcomes were lower with clomiphene; mortality was 1.83% versus 10.13%.

Participants / model
5,036 matched US veterans treated for hypogonadism
Treatment
Clomiphene citrate versus testosterone
Follow-up
Mean follow-up about 3.4 to 3.8 years
Study design
Retrospective administrative-database comparison

Infertility remained profoundly imbalanced (895 vs 41), and smoking, severity, medicines, symptoms, free testosterone, and bone density were omitted. The mortality contrast is not causal. Authors reported no funding or conflicts.

Read the original source
Bangladesh placebo RCT · semen outcomes

Randomized double-blind placebo-controlled trial

Hossain MJ, et al. Clinical and Experimental Reproductive Medicine. 2025. PMID 40899280. DOI 10.5653/cerm.2024.07353.

Among 46 analyzed men, clomiphene improved sperm concentration 9.17→13.88 million/mL, progressive motility 14.67%→21.42%, total motile count 3.53→7.81 million, and testosterone 372→806 ng/dL. Nausea occurred in two and dizziness in three.

Participants / model
50 eugonadal men with idiopathic oligoasthenozoospermia randomized; 46 analyzed
Treatment
Clomiphene citrate versus placebo
Follow-up
12 weeks
Study design
Single-center randomized double-blind placebo-controlled trial

No pregnancy or live-birth endpoint. The trial was registered after completion; funding was not stated and no relevant conflict was reported.

Read the original source
Pozzi et al. · 166-man sperm-response cohort

Retrospective cohort

Pozzi E, De Luca S, Birolini G, et al. World Journal of Men's Health. 2026. PMID 42533482. DOI 10.5534/wjmh.250371.

151/166 reached testosterone ≥3.5 ng/mL. Median sperm concentration rose 4.0→5.6 million/mL; 118 improved and 48 worsened by a median 3.3 million/mL.

Participants / model
166 hypogonadal oligospermic men
Treatment
Clomiphene citrate
Follow-up
At least 3 months; median follow-up 4 months
Study design
Single-center retrospective cohort

No comparator or pregnancy outcome, 11% dropout, exclusion of adverse-event discontinuations, and a white-European cohort limit inference. The authors reported no disclosure.

Read the original source
Ghanem et al. · clomiphene plus vitamin E

Randomized placebo-controlled combination trial

Ghanem H, Shaeer O, El-Segini A. Fertility and Sterility. 2010;93(7):2232-2235. PMID 19268928.

Pregnancy occurred in 11/30 couples assigned clomiphene plus vitamin E and 4/30 assigned placebo; OR 3.76 (95% CI 1.03 to 13.64).

Participants / model
60 men with idiopathic infertility and their partners
Treatment
Clomiphene plus vitamin E versus placebo
Follow-up
6 months
Study design
Randomized controlled combination-treatment trial

Vitamin E prevents attribution to clomiphene alone, and the confidence interval is wide.

Read the original source
Al Hashimi et al. · chosen mixed-treatment AAS cohort

Prospective nonrandomized comparative cohort

Al Hashimi M, et al. Andrologia. 2022. PMID 36065528. DOI 10.1111/and.14576.

After three months of observation, 463 of 520 former AAS users chose individualized treatment and 57 continued observation. Treated men recovered hormones, sexual function, testicular size, and semen earlier; 14 pregnancies were reported among 94 infertility presentations by month 12.

Participants / model
520 men after anabolic-androgenic steroid use
Treatment
Individualized hCG plus clomiphene, sometimes with tamoxifen, aromatase inhibitor, or FSH, versus observation
Follow-up
Up to 12 months after an initial 3-month observation period
Study design
Prospective cohort assigned by patient choice despite the paper's randomized label

No clomiphene-only arm. Baseline and treatment-selection confounding are severe. The paper inconsistently reports 74 versus 94 infertility cases. The authors reported no conflicts.

Read the original source
Henriksen et al. · mixed-intervention pilot

Open uncontrolled feasibility pilot

Henriksen HCB, et al. Performance Enhancement & Health. 2024;12(3):100283. DOI 10.1016/j.peh.2024.100283.

Of 81 screened and 17 eligible men, 10 completed. Five reached or ended within the normal testosterone range; withdrawal symptoms did not track testosterone response. Seven reported some clomiphene adverse effect at week 4, falling to three at week 16; no serious adverse event.

Participants / model
Men with long-term AAS use in substance-use-disorder care; 10 completers
Treatment
Clomiphene for all; six also received a short testosterone bridge and seven indicated hCG
Follow-up
16 weeks
Study design
Open uncontrolled feasibility pilot with mixed interventions
Funding
Public Norwegian and Oslo University Hospital support

Severe screening selection, co-treatment, clinical care, and time prevent clomiphene-only attribution.

Read the original source
İbis et al. · nonrandomized PCT cohort

Retrospective dual-center comparative cohort

İbis MA, et al. BJU International. Epub 2025. PMID 41147237. DOI 10.1111/bju.70059.

In 79 men, clomiphene-containing groups recovered hormones and semen earlier. All groups normalized hormones by month 6; at month 12 normozoospermia was 69.2% clomiphene, 87.5% clomiphene plus hCG, and 58.6% untreated.

Participants / model
79 recreational bodybuilders after no more than 6 months of AAS use with documented normal pre-cycle hormones and semen
Treatment
Observation, clomiphene, or clomiphene plus hCG; FSH suggested for five men
Follow-up
12 months
Study design
Retrospective nonrandomized dual-center cohort

Natural recovery was substantial, treatment was not randomized, adjusted estimates were imprecise, and there was no pregnancy or live-birth endpoint. Adverse-event and funding details remain unresolved.

Read the original source

Why is Clomiphene in A tier?

A for selected female ovulation induction, where randomized trials measured live birth. For men, clomiphene reliably changes hormones in selected patients, while symptom results are mixed, male-partner pregnancy benefit is unproved, post-AAS studies cannot isolate clomiphene, and no controlled healthy-performance trial was found.

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